Federica Gilardi

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59 publications

SMYD3: a new regulator of the early steps of adipocyte differentiation
Gilardi Federica, Sajic Tatjana, Gasser Marie, Caputo Tiziana, Bararpour Nasim, Augsburger Marc, Walter Nadia, Hainard Alexander, Fracasso Tony, Thomas Aurelien.
SMYD3: a new regulator of adipocyte precursor proliferation at the early steps of differentiation.
Sajic T., Ferreira Gomes C.K., Gasser M., Caputo T., Bararpour N., Landaluce-Iturriria E., Augsburger M., Walter N., Hainard A., Lopez-Mejia I.C. et al., 2024/04. International journal of obesity, 48 (4) pp. 557-566. Peer-reviewed.
Arsenic induces metabolome remodeling in mature human adipocytes.
Gasser M., Lenglet S., Bararpour N., Sajic T., Vaucher J., Wiskott K., Augsburger M., Fracasso T., Gilardi F., Thomas A., 2023/12. Toxicology, 500 p. 153672. Peer-reviewed.
Blood proteome of acute intracranial hemorrhage in infant victims of abusive head trauma.
Wiskott K., Gilardi F., Hainard A., Sanchez J.C., Thomas A., Sajic T., Fracasso T., 2023/02. Proteomics, 23 (3-4) pp. e2200078. Peer-reviewed.
Randomly controlled drivers using minimally invasive sampling: assessment of drug prevalence in Western Switzerland over two time periods.
Joye T., Déglon J., Donzé N., Gilardi F., Sidibé J., Favrat B., Augsburger M., Thomas A., 2022/12/28. BMC public health, 22 (1) p. 2446. Peer-reviewed.
 
Toxicity and Metabolomic Impact of Cobalt, Chromium, and Nickel Exposure on HepaRG Hepatocytes.
Bellouard M., Gasser M., Lenglet S., Gilardi F., Bararpour N., Augsburger M., Thomas A., Alvarez J.C., 2022/05/16. Chemical research in toxicology, 35 (5) pp. 807-816. Peer-reviewed.
 
A chemoinformatics search for peroxisome proliferator-activated receptors ligands revealed a new pan-agonist able to reduce lipid accumulation and improve insulin sensitivity.
Sblano S., Cerchia C., Laghezza A., Piemontese L., Brunetti L., Leuci R., Gilardi F., Thomas A., Genovese M., Santi A. et al., 2022/05/05. European journal of medicinal chemistry, 235 p. 114240. Peer-reviewed.
Creation of a Forensic Pathology Biobank in Switzerland: which issues and research opportunities?
Wiskott K., Gilardi F., Michaud K., Augsburger M., Castiglioni C., Carminati A., Grabherr S., Thomas A., Fracasso T., 2022/05. International journal of legal medicine, 136 (3) pp. 919-922. Peer-reviewed.
Cadmium acute exposure induces metabolic and transcriptomic perturbations in human mature adipocytes.
Gasser M., Lenglet S., Bararpour N., Sajic T., Wiskott K., Augsburger M., Fracasso T., Gilardi F., Thomas A., 2022/03/30. Toxicology, 470 p. 153153. Peer-reviewed.
Sex Dimorphism of Nonalcoholic Fatty Liver Disease (NAFLD) in Pparg-Null Mice.
Schiffrin M., Winkler C., Quignodon L., Naldi A., Trötzmüller M., Köfeler H., Henry H., Parini P., Desvergne B., Gilardi F., 2021/09/15. International journal of molecular sciences, 22 (18) p. 9969. Peer-reviewed.
Triangulating evidence from longitudinal and Mendelian randomization studies of metabolomic biomarkers for type 2 diabetes.
Porcu E., Gilardi F., Darrous L., Yengo L., Bararpour N., Gasser M., Marques-Vidal P., Froguel P., Waeber G., Thomas A. et al., 2021/03/18. Scientific reports, 11 (1) p. 6197. Peer-reviewed.
DBnorm as an R package for the comparison and selection of appropriate statistical methods for batch effect correction in metabolomic studies.
Bararpour N., Gilardi F., Carmeli C., Sidibe J., Ivanisevic J., Caputo T., Augsburger M., Grabherr S., Desvergne B., Guex N. et al., 2021/03/11. Scientific reports, 11 (1) p. 5657. Peer-reviewed.
Anti-adipogenic signals at the onset of obesity-related inflammation in white adipose tissue.
Caputo T., Tran VDT, Bararpour N., Winkler C., Aguileta G., Trang KB, Giordano Attianese GMP, Wilson A., Thomas A., Pagni M. et al., 2021/01. Cellular and molecular life sciences, 78 (1) pp. 227-247. Peer-reviewed.
Lack of Adiponectin Drives Hyperosteoclastogenesis in Lipoatrophic Mice.
Madel M.B., Fu H., Pierroz D.D., Schiffrin M., Winkler C., Wilson A., Pochon C., Toffoli B., Taïeb M., Jouzeau J.Y. et al., 2021. Frontiers in cell and developmental biology, 9 p. 627153. Peer-reviewed.
Identification of metabolomics biomarkers for type 2 diabetes: triangulating evidence from longitudinal and Mendelian randomization analyses
Porcu E., Gilardi F., Darrous L., Yengo L., Bararpour N., Gasser M., Vidal PM, Froguel P., Waeber G., Thomas A. et al., 2020/10/30..
Visualization and normalization of drift effect across batches in metabolome-wide association studies
Bararpour N., Gilardi F., Carmeli C., Sidibe J., Ivanisevic J., Caputo T., Augsburger M., Grabherr S., Desvergne B., Guex N. et al., 2020/01/22..
Systemic PPARγ deletion in mice provokes lipoatrophy, organomegaly, severe type 2 diabetes and metabolic inflexibility.
Gilardi F., Winkler C., Quignodon L., Diserens J.G., Toffoli B., Schiffrin M., Sardella C., Preitner F., Desvergne B., 2019/06. Metabolism, 95 pp. 8-20. Peer-reviewed.
Differential regulation of RNA polymerase III genes during liver regeneration.
Yeganeh M., Praz V., Carmeli C., Villeneuve D., Rib L., Guex N., Herr W., Delorenzi M., Hernandez N., CycliX consortium, 2019/02/28. Nucleic Acids Research, 47 (4) pp. 1786-1796. Peer-reviewed.
Renal mineralocorticoid receptor expression is reduced in lipoatrophy.
Toffoli B., Bernardi S., Winkler C., Carrascosa C., Gilardi F., Desvergne B., 2019/02. FEBS open bio, 9 (2) pp. 328-334. Peer-reviewed.
Cycles of gene expression and genome response during mammalian tissue regeneration.
Rib L., Villeneuve D., Minocha S., Praz V., Hernandez N., Guex N., Herr W., CycliX Consortium, 2018/09/12. Epigenetics & chromatin, 11 (1) p. 52. Peer-reviewed.
 
Delayed Hair Follicle Morphogenesis and Hair Follicle Dystrophy in a Lipoatrophy Mouse Model of Pparg Total Deletion.
Sardella C., Winkler C., Quignodon L., Hardman J.A., Toffoli B., Giordano Attianese GMP, Hundt J.E., Michalik L., Vinson C.R., Paus R. et al., 2018/03. The Journal of investigative dermatology, 138 (3) pp. 500-510. Peer-reviewed.
 
Hemicentin 1 influences podocyte dynamic changes in glomerular diseases.
Toffoli B., Zennaro C., Winkler C., Giordano Attianese GMP, Bernardi S., Carraro M., Gilardi F., Desvergne B., 2018. American Journal of Physiology. Renal physiology, 314 (6) pp. F1154-F1165. Peer-reviewed.
Lack of Adipocytes Alters Hematopoiesis in Lipodystrophic Mice.
Wilson A., Fu H., Schiffrin M., Winkler C., Koufany M., Jouzeau J.Y., Bonnet N., Gilardi F., Renevey F., Luther S.A. et al., 2018. Frontiers in immunology, 9 p. 2573. Peer-reviewed.
PPARγ Controls Ectopic Adipogenesis and Cross-Talks with Myogenesis During Skeletal Muscle Regeneration.
Dammone G., Karaz S., Lukjanenko L., Winkler C., Sizzano F., Jacot G., Migliavacca E., Palini A., Desvergne B., Gilardi F. et al., 2018. InternationalJjournal of Molecular Sciences, 19 (7) p. 2044. Peer-reviewed.
Will Widespread Synthetic Opioid Consumption Induce Epigenetic Consequences in Future Generations?
Gilardi F., Augsburger M., Thomas A., 2018. Frontiers in pharmacology, 9 p. 702. Peer-reviewed.
Diurnal regulation of RNA polymerase III transcription is under the control of both the feeding-fasting response and the circadian clock.
Mange F., Praz V., Migliavacca E., Willis I.M., Schütz F., Hernandez N., CycliX Consortium, 2017/06. Genome research, 27 (6) pp. 973-984. Peer-reviewed.
 
From chronic overnutrition to metaflammation and insulin resistance: adipose tissue and liver contributions.
Caputo T., Gilardi F., Desvergne B., 2017. FEBS Letters, 591 (19) pp. 3061-3088. Peer-reviewed.
HDAC3 is a molecular brake of the metabolic switch supporting white adipose tissue browning.
Ferrari A., Longo R., Fiorino E., Silva R., Mitro N., Cermenati G., Gilardi F., Desvergne B., Andolfo A., Magagnotti C. et al., 2017. Nature Communications, 8 (1) p. 93. Peer-reviewed.
Nephropathy in Pparg-null mice highlights PPARγ systemic activities in metabolism and in the immune system.
Toffoli B., Gilardi F., Winkler C., Soderberg M., Kowalczuk L., Arsenijevic Y., Bamberg K., Bonny O., Desvergne B., 2017. PLoS One, 12 (2) pp. e0171474. Peer-reviewed.
Transcriptional regulatory logic of the diurnal cycle in the mouse liver.
Sobel J.A., Krier I., Andersin T., Raghav S., Canella D., Gilardi F., Kalantzi A.S., Rey G., Weger B., Gachon F. et al., 2017. PLoS biology, 15 (4) pp. e2001069. Peer-reviewed.
 
Chlamydia pneumoniae acute liver infection affects hepatic cholesterol and triglyceride metabolism in mice.
Marangoni A., Fiorino E., Gilardi F., Aldini R., Scotti E., Nardini P., Foschi C., Donati M., Montagnani M., Cevenini M. et al., 2015/08. Atherosclerosis, 241 (2) pp. 471-479. Peer-reviewed.
 
Design, synthesis and biological evaluation of a class of bioisosteric oximes of the novel dual peroxisome proliferator-activated receptor α/γ ligand LT175.
Piemontese L., Fracchiolla G., Carrieri A., Parente M., Laghezza A., Carbonara G., Sblano S., Tauro M., Gilardi F., Tortorella P. et al., 2015. European Journal of Medicinal Chemistry, 90 pp. 583-594. Peer-reviewed.
Genome-wide analysis of SREBP1 activity around the clock reveals its combined dependency on nutrient and circadian signals.
Gilardi F., Migliavacca E., Naldi A., Baruchet M., Canella D., Le Martelot G., Guex N., Desvergne B., CycliX Consortium, 2014. PLoS Genetics, 10 (3) pp. e1004155. Peer-reviewed.
 
LT175 is a novel PPARα/γ ligand with potent insulin-sensitizing effects and reduced adipogenic properties.
Gilardi F., Giudici M., Mitro N., Maschi O., Guerrini U., Rando G., Maggi A., Cermenati G., Laghezza A., Loiodice F. et al., 2014. Journal of Biological Chemistry, 289 (10) pp. 6908-6920. Peer-reviewed.
Quantifying ChIP-seq data: a spiking method providing an internal reference for sample-to-sample normalization.
Bonhoure N., Bounova G., Bernasconi D., Praz V., Lammers F., Canella D., Willis I.M., Herr W., Hernandez N., Delorenzi M. et al., 2014. Genome Research, 24 (7) pp. 1157-1168. Peer-reviewed.
 
RXRs: collegial partners.
Gilardi F., Desvergne B., 2014. pp. 75-102 dans Asson-Batres M.A., Rochette-Egly C. (eds.) The biochemistry of retinoic acid receptors I: structure, activation, and function at the molecular level chap. 5, Springer.
 
Inflammatory serum proteome pattern in mice fed a high-fat diet.
Gianazza E., Sensi C., Eberini I., Gilardi F., Giudici M., Crestani M., 2013/03. Amino acids, 44 (3) pp. 1001-1008. Peer-reviewed.
Inhibition of class I histone deacetylases unveils a mitochondrial signature and enhances oxidative metabolism in skeletal muscle and adipose tissue.
Galmozzi A., Mitro N., Ferrari A., Gers E., Gilardi F., Godio C., Cermenati G., Gualerzi A., Donetti E., Rotili D. et al., 2013. Diabetes, 62 (3) pp. 732-742. Peer-reviewed.
 
Molecular determinants for nuclear receptors selectivity: chemometric analysis, dockings and site-directed mutagenesis of dual peroxisome proliferator-activated receptors α/γ agonists.
Carrieri A., Giudici M., Parente M., De Rosas M., Piemontese L., Fracchiolla G., Laghezza A., Tortorella P., Carbonara G., Lavecchia A. et al., 2013. European Journal of Medicinal Chemistry, 63 pp. 321-332. Peer-reviewed.
 
Site-Directed Mutagenesis to Study the Role of Specific Amino Acids in the Ligand Binding Domain of PPARs
Mitro Nico, Gilardi Federica, Giudici Marco, Godio Cristina, Scotti Elena, Crestani Maurizio, 2013. pp. 137-144 dans Peroxisome Proliferator-Activated Receptors (PPARs), Humana Press.
 
SOCS3 Transactivation by PPARγ Prevents IL-17-Driven Cancer Growth.
Berger H., Végran F., Chikh M., Gilardi F., Ladoire S., Bugaut H., Mignot G., Chalmin F., Bruchard M., Derangère V. et al., 2013. Cancer Research, 73 (12) pp. 3578-3590. Peer-reviewed.
 
Synthesis, characterization and biological evaluation of ureidofibrate-like derivatives endowed with peroxisome proliferator-activated receptor activity.
Porcelli L., Gilardi F., Laghezza A., Piemontese L., Mitro N., Azzariti A., Altieri F., Cervoni L., Fracchiolla G., Giudici M. et al., 2012/01/12. Journal of medicinal chemistry, 55 (1) pp. 37-54. Peer-reviewed.
A multiplicity of factors contributes to selective RNA polymerase III occupancy of a subset of RNA polymerase III genes in mouse liver.
Canella D., Bernasconi D., Gilardi F., LeMartelot G., Migliavacca E., Praz V., Cousin P., Delorenzi M., Hernandez N., CycliX Consortium, 2012. Genome Research, 22 (4) pp. 666-680. Peer-reviewed.
Genome-wide RNA polymerase II profiles and RNA accumulation reveal kinetics of transcription and associated epigenetic changes during diurnal cycles.
Le Martelot G., Canella D., Symul L., Migliavacca E., Gilardi F., Liechti R., Martin O., Harshman K., Delorenzi M., Desvergne B. et al., 2012. PLoS Biology, 10 (11) pp. e1001442. Peer-reviewed.
 
Linking epigenetics to lipid metabolism: focus on histone deacetylases.
Ferrari A., Fiorino E., Giudici M., Gilardi F., Galmozzi A., Mitro N., Cermenati G., Godio C., Caruso D., De Fabiani E. et al., 2012. Molecular Membrane Biology, 29 (7) pp. 257-266. Peer-reviewed.
 
Structural insight into peroxisome proliferator-activated receptor gamma binding of two ureidofibrate-like enantiomers by molecular dynamics, cofactor interaction analysis, and site-directed mutagenesis.
Pochetti G., Mitro N., Lavecchia A., Gilardi F., Besker N., Scotti E., Aschi M., Re N., Fracchiolla G., Laghezza A. et al., 2010/06/10. Journal of medicinal chemistry, 53 (11) pp. 4354-4366. Peer-reviewed.
 
When food meets man: the contribution of epigenetics to health.
De Fabiani E., Mitro N., Gilardi F., Galmozzi A., Caruso D., Crestani M., 2010/05. Nutrients, 2 (5) pp. 551-571. Peer-reviewed.
 
Olive oil phenols modulate the expression of metalloproteinase 9 in THP-1 cells by acting on nuclear factor-kappaB signaling.
Dell'Agli M., Fagnani R., Galli G.V., Maschi O., Gilardi F., Bellosta S., Crestani M., Bosisio E., De Fabiani E., Caruso D., 2010/02/24. Journal of agricultural and food chemistry, 58 (4) pp. 2246-2252. Peer-reviewed.
 
Sterol–Protein Interactions in Cholesterol and Bile Acid Synthesis
De Fabiani Emma, Mitro Nico, Gilardi Federica, Crestani Maurizio, 2010. pp. 109-135 dans Cholesterol Binding and Cholesterol Transport Proteins:, Springer Netherlands.
 
Expression of sterol 27-hydroxylase in glial cells and its regulation by liver X receptor signaling.
Gilardi F., Viviani B., Galmozzi A., Boraso M., Bartesaghi S., Torri A., Caruso D., Crestani M., Marinovich M., de Fabiani E., 2009/12/01. Neuroscience, 164 (2) pp. 530-540. Peer-reviewed.
 
Crystal structure of the peroxisome proliferator-activated receptor gamma (PPARgamma) ligand binding domain complexed with a novel partial agonist: a new region of the hydrophobic pocket could be exploited for drug design.
Montanari R., Saccoccia F., Scotti E., Crestani M., Godio C., Gilardi F., Loiodice F., Fracchiolla G., Laghezza A., Tortorella P. et al., 2008/12/25. Journal of medicinal chemistry, 51 (24) pp. 7768-7776. Peer-reviewed.
 
Bile acids and gene regulation: from nuclear receptors to chromatin.
Mitro N., Gilardi F., Godio C., Scotti E., De Fabiani E., Caruso D., Crestani M., 2008/05/01. Frontiers in bioscience, 13 pp. 6276-6288. Peer-reviewed.
 
The pharmacological exploitation of cholesterol 7alpha-hydroxylase, the key enzyme in bile acid synthesis: from binding resins to chromatin remodelling to reduce plasma cholesterol.
Gilardi F., Mitro N., Godio C., Scotti E., Caruso D., Crestani M., De Fabiani E., 2007/12. Pharmacology & therapeutics, 116 (3) pp. 449-472. Peer-reviewed.
 
Bile acids and their signaling pathways: eclectic regulators of diverse cellular functions.
Scotti E., Gilardi F., Godio C., Gers E., Krneta J., Mitro N., De Fabiani E., Caruso D., Crestani M., 2007/10. Cellular and molecular life sciences, 64 (19-20) pp. 2477-2491. Peer-reviewed.
 
Insights in the regulation of cholesterol 7alpha-hydroxylase gene reveal a target for modulating bile acid synthesis.
Mitro N., Godio C., De Fabiani E., Scotti E., Galmozzi A., Gilardi F., Caruso D., Vigil Chacon A.B., Crestani M., 2007/09. Hepatology, 46 (3) pp. 885-897. Peer-reviewed.
 
Molecular mechanisms underlying mancozeb-induced inhibition of TNF-alpha production.
Corsini E., Viviani B., Birindelli S., Gilardi F., Torri A., Codecà I., Lucchi L., Bartesaghi S., Galli C.L., Marinovich M. et al., 2006/04/15. Toxicology and applied pharmacology, 212 (2) pp. 89-98. Peer-reviewed.
 
Bile acid signaling to the nucleus: finding new connections in the transcriptional regulation of metabolic pathways.
De Fabiani E., Mitro N., Godio C., Gilardi F., Caruso D., Crestani M., 2004/11. Biochimie, 86 (11) pp. 771-778. Peer-reviewed.
 
LXR (liver X receptor) and HNF-4 (hepatocyte nuclear factor-4): key regulators in reverse cholesterol transport.
Crestani M., De Fabiani E., Caruso D., Mitro N., Gilardi F., Vigil Chacon A.B., Patelli R., Godio C., Galli G., 2004/02. Biochemical Society transactions, 32 (Pt 1) pp. 92-96. Peer-reviewed.
 
Coordinated control of cholesterol catabolism to bile acids and of gluconeogenesis via a novel mechanism of transcription regulation linked to the fasted-to-fed cycle.
De Fabiani E., Mitro N., Gilardi F., Caruso D., Galli G., Crestani M., 2003/10/03. The Journal of biological chemistry, 278 (40) pp. 39124-39132. Peer-reviewed.
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